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Home > Category > > Small Molecule Compound > VU0134992 hydrochloride

VU0134992 hydrochloride

Glpbio
Catalog No:GC39667-10mM (in 1mL DMSO) CAS No.:1052515-91-9 MDLNo: Brand:Glpbio purity: 特性: Purpose:VU0134992 hydrochloride 是第一個(gè)亞型偏好的,具有口服活性和選擇性的內(nèi)向整流鉀通道 Kir4.1 阻滯劑,IC50 值為 0.97 μM。VU0134992 hydrochloride 在 -120 mV 時(shí),對同分 Kir4.1 比 Kir4.1/5.1 共分通道 (IC50=9 μM) 高出 9 倍的選擇性。DMSO: 250 mg/mL (558.24 mM)
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